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SB 742457
CAS No. 607742-69-8
SB 742457 ( GSK742457 )
Catalog No. M15279 CAS No. 607742-69-8
SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 61 | In Stock |
|
| 10MG | 98 | In Stock |
|
| 25MG | 200 | In Stock |
|
| 50MG | 320 | In Stock |
|
| 100MG | 507 | In Stock |
|
| 500MG | 1062 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSB 742457
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NoteResearch use only, not for human use.
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Brief DescriptionSB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.
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DescriptionSB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63, exhibits >100-fold selectivity over other receptors. Phase 2.
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SynonymsGSK742457
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT6
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number607742-69-8
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Formula Weight353.44
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Molecular FormulaC19H19N3O2S
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Purity>98%(HPLC)
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SolubilityEthanol: 2 mg/mL (5.65 mM); DMSO: 78 mg/mL (220.68 mM)
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SMILESO=S(C1=CC2=CC=CC(N3CCNCC3)=C2N=C1)(C4=CC=CC=C4)=O
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Chemical Name3-Phenylsulfonyl-8-(piperazin-1-yl)quinoline
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Chuang ATT, et al. Alzheimers Dement, 2006, 2, S631–S632 (abstract).
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